L. ANGEL

Evidence from opiate binding studies that heroin acts through its metabolites

Charles E. Inturrisi, Michael Schultz, Sang J. Shin et al. · Life Sciences · 1983 · 211 citations

Opioid Epidemic, Substance Abuse, Substance Use +10

Multiple Opiate Receptors: Alcohol Selectively Inhibits Binding to Delta Receptors

Jacob M. Hiller, L. ANGEL, Eric J. Simon · Science · 1981 · 148 citations

Characterization of the selective inhibition of the delta subclass of opioid binding sites by alcohols.

J M Hiller, L. ANGEL, Eric J. Simon · Molecular Pharmacology · 1984 · 27 citations

Quaternary derivatives of narcotic antagonists: Stereochemical requirements at the chiral nitrogen for and activity

Angelo Bianchetti, Dino Nisato, R. Sacilotto et al. · Life Sciences · 1983 · 22 citations

Pharmaceutical Chemistry, Biochemistry, Medicine +8

Diastereomeric 6-desoxy-6-spiro-.alpha.-methylene-.gamma.-butyrolactone derivatives of naltrexone and oxymorphone. Selective irreversible inhibition of naltrexone binding in an opioid receptor preparation by a conformationally restricted Michael acceptor ligand

Gary A. Koolpe, Wendel L. Nelson, Theresa L. Gioannini et al. · Journal of Medicinal Chemistry · 1984 · 11 citations · Full text

Bioorganic Chemistry, Diastereomeric 6-Desoxy-6-spiro-.alpha.-methylene-.gamma.-butyrolactone, Organic Chemistry +22