Gianni Casaluce

Toward the Discovery of Novel Anti‐HIV Drugs. Second‐Generation Inhibitors of the Cellular ATPase DDX3 with Improved Anti‐HIV Activity: Synthesis, Structure–Activity Relationship Analysis, Cytotoxicity Studies, and Target Validation

Giovanni Maga, Federico Falchi, Marco Radi et al. · ChemMedChem · 2011 · 105 citations

Practical One-Pot Two-Step Protocol for the Microwave-Assisted Synthesis of Highly Functionalized Rhodanine Derivatives

Marco Radi, Lorenzo Botta, Gianni Casaluce et al. · Journal of Combinatorial Chemistry · 2009 · 58 citations

Discovery of Chiral Cyclopropyl Dihydro-Alkylthio-Benzyl-Oxopyrimidine (<i>S</i>-DABO) Derivatives as Potent HIV-1 Reverse Transcriptase Inhibitors with High Activity Against Clinically Relevant Mutants

Marco Radi, Giovanni Maga, Maddalena Alongi et al. · Journal of Medicinal Chemistry · 2009 · 38 citations · Full text

Synthesis, Biological Activity, and ADME Properties of Novel <i>S</i>‐DABOs/<i>N</i>‐DABOs as HIV Reverse Transcriptase Inhibitors

Marco Radi, Mafalda Pagano, Luigi Franchi et al. · ChemMedChem · 2012 · 13 citations