Thomas Leiser

Defining the Mechanism of Action and Enzymatic Selectivity of Psammaplin A against Its Epigenetic Targets

Matthias G. J. Baud, Thomas Leiser, Patricia Haus et al. · Journal of Medicinal Chemistry · 2012 · 96 citations · Full text

Drug Target, Epigenetic Change, Molecular Biology +20

Thioester derivatives of the natural product psammaplin A as potent histone deacetylase inhibitors

Matthias G. J. Baud, Thomas Leiser, Vanessa Petrucci et al. · Beilstein Journal of Organic Chemistry · 2013 · 30 citations · Full text

Thioester Derivatives, Medicinal Chemistry, Derivative (Chemistry) +15

New synthetic strategies towards psammaplin A, access to natural product analogues for biological evaluation

Matthias G. J. Baud, Thomas Leiser, Franz‐Josef Meyer‐Almes et al. · Organic & Biomolecular Chemistry · 2010 · 29 citations

Bioorganic Chemistry, A Analogues, Pharmaceutical Chemistry +17

Highly Ligand Efficient and Selective <i>N</i>‐2‐(Thioethyl)picolinamide Histone Deacetylase Inhibitors Inspired by the Natural Product Psammaplin A

Matthias G. J. Baud, Patricia Haus, Thomas Leiser et al. · ChemMedChem · 2012 · 19 citations