Concepedia
Statistics
Publications
8
Citations
234
H-Index
Active since
2016
Affiliations
Université de Lille(Current)
Inserm
Lille Inflammation Research International Center
Alexandru Ioan Cuza University
Hautes Études d'Ingénieur
Germain Homerin is an author at Université de Lille specializing in pharmacology, medicinal chemistry, and drug discovery.
Publications per year
2016–2021
A small-molecule P2RX7 activator promotes anti-tumor immune responses and sensitizes lung tumor to immunotherapy
Laëtitia Douguet, Séréna Janho dit Hreich, Jonathan Benzaquen et al. · Nature Communications · 2021 · 91 citations · Full text
Medicine, Oncology, Pharmacology +17
Pyroglutamide-Based P2X7 Receptor Antagonists Targeting Inflammatory Bowel Disease
Germain Homerin, Samir Jawhara, Xavier Dezitter et al. · Journal of Medicinal Chemistry · 2019 · 42 citations · Full text
Medicine, Medicinal Chemistry, Pharmacology +17
Studies on phenothiazines: New microtubule-interacting compounds with phenothiazine A-ring as potent antineoplastic agents
Alina Ghinet, Iuliana-Monica Moise, Germain Homerin et al. · Bioorganic & Medicinal Chemistry · 2016 · 31 citations · Full text
Medicine, Medicinal Chemistry, Pharmacology +12
ZrCl4 as a new catalyst for ester amidation: an efficient synthesis of h-P2X7R antagonists
Germain Homerin, Davy Baudelet, Pierrick Dufrénoy et al. · Tetrahedron Letters · 2016 · 18 citations
Natural Sciences, Chemistry, Medicinal Chemistry +9
On the discovery of new potent human farnesyltransferase inhibitors: emerging pyroglutamic derivatives
Germain Homerin, Emmanuelle Lipka, Amaury Farce et al. · Organic & Biomolecular Chemistry · 2017 · 15 citations
Pharmacy, Medicinal Chemistry, Pharmacology +10
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