Pharmacological profile of LF 16-0687, a new potent non-peptide bradykinin B2 receptor antagonist

Didier Pruneau, Jean Luc Paquet, J.M. Luccarini, +9

Immunopharmacology

BiochemistryMedicinePeptide LibraryNeuropeptide ReceptorPharmacotherapy +5

Characterization of the molecular interactions of interleukin-8 (CXCL8), growth related oncogen α (CXCL1) and a non-peptide antagonist (SB 225002) with the human CXCR2

Julie Catusse, Anne Liotard, Bruno Loillier, +2

Biochemical Pharmacology

InflammationCytokineMolecular ImmunologyHuman Cxcr2Sb 225002 +10

Stable expression of human kinin B₁ receptor in 293 cells: pharmacological and functional characterization

S. Bastian, Bruno Loillier, J L Paquet, +1

British Journal of Pharmacology

Molecular RegulationDissociation ConstantImmunologyCellular PharmacologyBinding Properties +17

Haemodynamic and cardiac effects of kinin B₁ and B₂ receptor stimulation in conscious instrumented dogs

Pierre Bélichard, Bruno Loillier, Jean Luc Paquet, +2

British Journal of Pharmacology

Cardiac EffectsConscious Instrumented DogsNitric OxideBradykinin B1Cardiovascular Pharmacology +20

LF 16.0335, a novel potent and selective nonpeptide antagonist of the human bradykinin B₂ receptor

Didier Pruneau, Jean‐Michel Luccarini, Chantal Fouchet, +8

British Journal of Pharmacology

Molecular PharmacologyMolecular PhysiologyLf 16.0335BiochemistryMedicine +13

Pharmacological characterization of the bradykinin B₂ receptor: inter‐species variability and dissociation between binding and functional responses

J L Paquet, J.M. Luccarini, Chantal Fouchet, +6

British Journal of Pharmacology

Identification of a Key Region of Kinin B1 Receptor for High Affinity Binding of Peptide Antagonists

S. Bastian, Didier Pruneau, Bruno Loillier, +3

Journal of Biological Chemistry

Interleukin 8 (IL-8) Induces the Expression of Kinin B1Receptor in Human Lung Fibroblasts

S. Bastian, J L Paquet, Claude Robert, +6

Biochemical and Biophysical Research Communications

InflammationKinin B1receptorCytokineInflammatory Lung DiseaseLung Inflammation +8

Cloning and characterization of guinea pig interleukin-8 receptor

Julie Catusse, Patrick Faye, Bruno Loillier, +5

Biochemical Pharmacology

InflammationCytokineImmunologyAutoimmunityMedicine

In vitro and in vivo effects of the new nonpeptide bradykinin B₂receptor antagonist, LF 16‐0335C, on guinea‐pig and rat kinin receptors

Didier Pruneau, Jean‐Michel Luccarini, Chantal Fouchet, +8

Fundamental and Clinical Pharmacology