Strain-release amination

Ryan Gianatassio, Justin M. Lopchuk, Jie Wang, +11

Science

Combinatorial ChemistryMedicinal ChemistryBioorganic ChemistryDrug CandidatesBiochemistry +9

Functionalized olefin cross-coupling to construct carbon–carbon bonds

Julian C. Lo, Jinghan Gui, Yuki Yabe, +2

Nature

Materials ScienceCross-coupling ReactionEngineeringCovalent Bonded FrameworkOrganic Chemistry +2

Strain-Release Heteroatom Functionalization: Development, Scope, and Stereospecificity

Justin M. Lopchuk, Kasper Fjelbye, Yu Kawamata, +21

Journal of the American Chemical Society

Palau’chlor: A Practical and Reactive Chlorinating Reagent

Rodrigo A. Rodriguez, Chung‐Mao Pan, Yuki Yabe, +3

Journal of the American Chemical Society

Diversity Oriented SynthesisEngineeringHeterocyclicNatural SciencesDiversity-oriented Synthesis +10

C–H Methylation of Heteroarenes Inspired by Radical SAM Methyl Transferase

Jinghan Gui, Qianghui Zhou, Chung‐Mao Pan, +6

Journal of the American Chemical Society

Combinatorial ChemistryEngineeringZinc BisSimple ProtocolMolecular Biology +16

Bioconjugation by Native Chemical Tagging of C–H Bonds

Qianghui Zhou, Jinghan Gui, Chung‐Mao Pan, +6

Journal of the American Chemical Society

Design and synthesis of Hsp90 inhibitors: Exploring the SAR of Sansalvamide A derivatives

Robert P. Sellers, Leslie D. Alexander, Victoria A. Johnson, +13

Bioorganic & Medicinal Chemistry

Sansalvamide A DerivativesMedicinal ChemistryPharmaceutical ScienceDerivativesHsp90 Inhibitors +10

Synthesis of Second-Generation Sansalvamide A Derivatives: Novel Templates as Potential Antitumor Agents

Rodrigo A. Rodriguez, Po‐Shen Pan, Chung‐Mao Pan, +9

The Journal of Organic Chemistry

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A comprehensive study of Sansalvamide A derivatives: The structure–activity relationships of 78 derivatives in two pancreatic cancer cell lines

Po‐Shen Pan, Robert C. Vasko, Stephanie A. Lapera, +7

Bioorganic & Medicinal Chemistry

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Synthesis of Sansalvamide A derivatives and their cytotoxicity in the MSS colon cancer cell line HT-29

Thomas J. Styers, Ahmet Kekec, Rodrigo A. Rodriguez, +12

Bioorganic & Medicinal Chemistry

Sansalvamide A DerivativesMedicinal ChemistryMedicineAnti-cancer AgentDrug Development +3