Synthesis and antitumor activity of 2,5-bis(3′-indolyl)-furans and 3,5-bis(3′-indolyl)-isoxazoles, nortopsentin analogues

Patrizia Diana, Anna Carbone, Paola Barraja, +3

Bioorganic & Medicinal Chemistry

Medicinal ChemistryNatural SciencesMedicineOrganic ChemistryNortopsentin Analogues +5

Chemistry, antiproliferative properties, tumor selectivity, and molecular mechanisms of novel gold(III) compounds for cancer treatment: a systematic study

Angela Casini, Gerhard Kelter, Chiara Gabbiani, +5

JBIC Journal of Biological Inorganic Chemistry

Medicinal ChemistryNovel GoldMetal NanoparticlesMedicineNatural Sciences +8

Mansouramycins A−D, Cytotoxic Isoquinolinequinones from a Marine Streptomycete

Usama W. Hawas, Mohamed Shaaban, Khaled A. Shaaban, +7

Journal of Natural Products

Role of Transferrin Receptor and the ABC Transporters ABCB6 and ABCB7 for Resistance and Differentiation of Tumor Cells towards Artesunate

Gerhard Kelter, Daniel Steinbach, V. Badireenath Konkimalla, +4

PLoS ONE

Chemoprevention StrategyIron MetabolismRedox BiologyCellular PhysiologyTumor Biology +17

In-vitro anti-tumor activity studies of bridged and unbridged benzyl-substituted titanocenes

Gerhard Kelter, Nigel J. Sweeney, Katja Strohfeldt, +2

Anti-Cancer Drugs

Organic ChemistryChemistryHeterocycle ChemistryTumor BiologyMedicinal Chemistry +18

Antitumor Activity of Bis-indole Derivatives

Aldo Andreani, Silvia Burnelli, Massimiliano Granaiola, +13

Journal of Medicinal Chemistry

Proteasome InhibitionMedicinal ChemistryBiochemistryMedicineNatural Sciences +9

Lung Cancer: EGFR Inhibitors with Low Nanomolar Activity against a Therapy‐Resistant L858R/T790M/C797S Mutant

Marcel Günther, Michael Juchum, Gerhard Kelter, +2

Angewandte Chemie International Edition

Drug TargetingOncologyNovel TherapyTumor MicroenvironmentMedicine +13

Epoxyphomalin A and B, Prenylated Polyketides with Potent Cytotoxicity from the Marine-Derived Fungus <i>Phoma</i> sp.

Ietidal E. Mohamed, Harald Gross, Alexander Pontius, +6

Organic Letters

Bioorganic ChemistryMedicinal FungiPrenylated PolyketidesMedicinal ChemistryUnusual Structural Features +14

N -heterocyclic carbenes (NHC) with 1,2,4-oxadiazole-substituents related to natural products: Synthesis, structure and potential antitumor activity of some corresponding gold(I) and silver(I) complexes

Catalin V. Maftei, Elena Fodor, Peter G. Jones, +6

European Journal of Medicinal Chemistry

Inorganic ChemistryMedicinal ChemistryEngineeringHeterocyclicNatural Sciences +10

Anticancer Properties of Distinct Antimalarial Drug Classes

Rob Hooft van Huijsduijnen, R. Kiplin Guy, Kelly Chibale, +7

PLoS ONE

Antiparasitic AgentMalariaDhfr InhibitorsPharmaceutical ChemistryMolecular Pharmacology +15