Natacha Novosad

Design, Synthesis and Biological Evaluation of 4‐Amino‐<i>N</i>‐(4‐aminophenyl)benzamide Analogues of Quinoline‐Based SGI‐1027 as Inhibitors of DNA Methylation

Elodie Rilova, Alexandre Erdmann, Christina Gros et al. · ChemMedChem · 2014 · 67 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +15

Rational Design of Bisubstrate-Type Analogues as Inhibitors of DNA Methyltransferases in Cancer Cells

Ludovic Halby, Yoann Menon, Elodie Rilova et al. · Journal of Medicinal Chemistry · 2017 · 59 citations · Full text

Medicine, Medicinal Chemistry, Oncology +16

Design and synthesis of new non nucleoside inhibitors of DNMT3A

Alexandre Erdmann, Yoann Menon, Christina Gros et al. · Bioorganic & Medicinal Chemistry · 2015 · 25 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +8

Consequences of combining siRNA-mediated DNA methyltransferase 1 depletion with 5-aza-2′-deoxycytidine in human leukemic KG1 cells

Stéphane Vispé, Arthur Deroide, Emeline Davoine et al. · Oncotarget · 2015 · 16 citations · Full text

Life Sciences, Molecular Biology, Oncology +14

Identification and Optimization of Hydrazone-Gallate Derivatives as Specific Inhibitors of DNA Methyltransferase 3A

Alexandre Erdmann, Yoann Menon, Christina Gros et al. · Future Medicinal Chemistry · 2016 · 16 citations

Pharmacy, Medicinal Chemistry, Pharmacology +14