Paul Gaspari

Structure−Activity Study of Brassinin Derivatives as Indoleamine 2,3-Dioxygenase Inhibitors

Paul Gaspari, Tinku Banerjee, William P. Malachowski et al. · Journal of Medicinal Chemistry · 2005 · 179 citations · Full text

A key in vivo antitumor mechanism of action of natural product-based brassinins is inhibition of indoleamine 2,3-dioxygenase

Tinku Banerjee, James B. DuHadaway, Paul Gaspari et al. · Oncogene · 2007 · 172 citations · Full text

Medicinal Chemistry, Biochemistry, Natural Product-based Brassinins +11

Asymmetric Synthesis of Acyclic 1,3-Amino Alcohols by Reduction of <i>N</i>-Sulfinyl β-Amino Ketones. Formal Synthesis of (−)-Pinidinol and (+)- Epipinidinol

Franklin A. Davis, Paul Gaspari, Brad M. Nolt et al. · The Journal of Organic Chemistry · 2008 · 70 citations

Rational design of novel, potent piperazinone and imidazolidinone BACE1 inhibitors

Jared N. Cumming, Thuy X. Le, Sethu Geetha Babu et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 58 citations · Full text

Medicinal Chemistry, Biochemistry, Drug Design +11

Asymmetric Synthesis of Substituted Tropinones Using the Intramolecular Mannich Cyclization Reaction and Acyclic <i>N</i>-Sulfinyl β-Amino Ketone Ketals

Franklin A. Davis, Naresh Theddu, Paul Gaspari · Organic Letters · 2009 · 33 citations · Full text