Dario Masullo

Modification on Ursodeoxycholic Acid (UDCA) Scaffold. Discovery of Bile Acid Derivatives As Selective Agonists of Cell-Surface G-Protein Coupled Bile Acid Receptor 1 (GP-BAR1)

Valentina Sepe, Barbara Renga, Carmen Festa et al. · Journal of Medicinal Chemistry · 2014 · 90 citations · Full text

Molecular Pharmacology, Molecular Physiology, Biochemistry +14

Insights on FXR selective modulation. Speculation on bile acid chemical space in the discovery of potent and selective agonists

Valentina Sepe, Carmen Festa, Barbara Renga et al. · Scientific Reports · 2016 · 47 citations · Full text

Hyodeoxycholic acid derivatives as liver X receptor α and G-protein-coupled bile acid receptor agonists

Simona De Marino, Adriana Carino, Dario Masullo et al. · Scientific Reports · 2017 · 42 citations · Full text

Zn-Catalyzed Nicotinate-Directed Transamidations in Peptide Synthesis

Charlie Hollanders, Evelien Renders, Charlène Gadais et al. · ACS Catalysis · 2020 · 27 citations

Combinatorial Chemistry, Biochemistry, Zn-catalyzed Nicotinate-directed Transamidations +12

Investigation on bile acid receptor regulators. Discovery of cholanoic acid derivatives with dual G-protein coupled bile acid receptor 1 (GPBAR1) antagonistic and farnesoid X receptor (FXR) modulatory activity

Valentina Sepe, Barbara Renga, Carmen Festa et al. · Steroids · 2015 · 19 citations

Molecular Pharmacology, Biochemistry, Biliary Tract +9