Holger Kubas

Multivalent cyclic RGD ligands: influence of linker lengths on receptor binding

Holger Kubas, Martin Schäfer, Ulrike Bauder‐Wüst et al. · Nuclear Medicine and Biology · 2010 · 42 citations

Molecular Docking, Signal Transduction, Biochemistry +11

The effect of buffer species on biorelevant dissolution and precipitation assays – Comparison of phosphate and bicarbonate buffer

Katharina Krollik, Andreas Lehmann, Christian Wagner et al. · European Journal of Pharmaceutics and Biopharmaceutics · 2021 · 32 citations

Bioconcentration, Organic Geochemistry, Environmental Chemistry +8

Improved Prediction of in Vivo Supersaturation and Precipitation of Poorly Soluble Weakly Basic Drugs Using a Biorelevant Bicarbonate Buffer in a Gastrointestinal Transfer Model

Christian Jede, Christian Wagner, Holger Kubas et al. · Molecular Pharmaceutics · 2019 · 30 citations

In-line derivative spectroscopy as a promising application to a small-scale <i>in vitro</i> transfer model in biorelevant supersaturation and precipitation testing

Christian Jede, Christian Wagner, Holger Kubas et al. · Journal of Pharmacy and Pharmacology · 2018 · 16 citations

Scaffold hopping approach towards various AFQ-056 analogs as potent metabotropic glutamate receptor 5 negative allosteric modulators

Holger Kubas, Udo Meyer, Mirko Hechenberger et al. · Bioorganic & Medicinal Chemistry Letters · 2013 · 14 citations · Full text

Negative Allosteric Modulators, Biochemistry, Functional Selectivity +6