Gameel A. M. Elhagali

<i>In Vitro</i> Antimicrobial Evaluation, Single-Point Resistance Study, and Radiosterilization of Novel Pyrazole Incorporating Thiazol-4-one/Thiophene Derivatives as Dual DNA Gyrase and DHFR Inhibitors against MDR Pathogens

Hazem Ali Mohamed, Yousry A. Ammar, Gameel A. M. Elhagali et al. · ACS Omega · 2022 · 68 citations · Full text

Synthesis, characterization, and in vitro antibacterial activity of some new pyridinone and pyrazole derivatives with some in silico ADME and molecular modeling study

Khadija E. Saadon, Nadia M. H. Taha, N. A. Mahmoud et al. · Journal of the Iranian Chemical Society · 2022 · 64 citations · Full text

Cyanoacrylamide Derivatives, Engineering, Organic Chemistry +21

A new exploration toward adamantane derivatives as potential anti‐MDR agents: Design, synthesis, antimicrobial, and radiosterilization activity as potential topoisomerase IV and DNA gyrase inhibitors

Ahmed Ragab, Moustafa S. Abusaif, Dina S. Aboul‐Magd et al. · Drug Development Research · 2022 · 51 citations

Discovery a novel of thiazolo[3,2-a]pyridine and pyrazolo[3,4-d]thiazole derivatives as DNA gyrase inhibitors; design, synthesis, antimicrobial activity, and some in-silico ADMET with molecular docking study

Hazem Ali Mohamed, Yousry A. Ammar, Gameel A. M. Elhagali et al. · Journal of Molecular Structure · 2023 · 44 citations

Medicinal Chemistry, Biochemistry, Medicine +9

Hybridized Quinoline Derivatives as Anticancer Agents: Design, Synthesis, Biological Evaluation and Molecular Docking

Mohamed R. Selim, M. A. Zahran, Amany Belal et al. · Anti-Cancer Agents in Medicinal Chemistry · 2018 · 36 citations

Combinatorial Chemistry, Pharmaceutical Science, Bioorganic Chemistry +18