Concepedia

Discovery a novel of thiazolo[3,2-a]pyridine and pyrazolo[3,4-d]thiazole derivatives as DNA gyrase inhibitors; design, synthesis, antimicrobial activity, and some in-silico ADMET with molecular docking study

Hazem Ali Mohamed, Yousry A. Ammar, Gameel A. M. Elhagali, Hassan A. Eyada, Dina S. Aboul‐Magd, Ahmed Ragab

Journal of Molecular Structure · 2023 · 44 citations · 52 references

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References

52

Dihydropyrimidine calcium channel blockers: 2-heterosubstituted 4-aryl-1,4-dihydro-6-methyl-5-pyrimidinecarboxylic acid esters as potent mimics of dihydropyridines

Karnail S. Atwal, George C. Rovnyak, Joseph E. Schwartz et al. · Journal of Medicinal Chemistry · 1990 · 284 citations · Full text

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Design, synthesis, computational and biological evaluation of new anxiolytics

Athina Geronikaki, John C. Dearden, Wim Dehaen et al. · Bioorganic & Medicinal Chemistry · 2004 · 135 citations · Full text

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Green chemoselective synthesis of thiazolo[3,2-a]pyridine derivatives and evaluation of their antioxidant and cytotoxic activities

Feng Shi, Chunmei Li, Ming Xia et al. · Bioorganic & Medicinal Chemistry Letters · 2009 · 118 citations

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Synthesis and antiviral activity of some new bis-1,3-thiazole derivatives

Kamal M. Dawood, Taha M. A. Eldebss, Heba S. A. Elzahabi et al. · European Journal of Medicinal Chemistry · 2015 · 111 citations

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Synthesis, anti-inflammatory and anti-ulcer evaluations of thiazole, thiophene, pyridine and pyran derivatives derived from androstenedione

Rafat M. Mohareb, Mayssoune Y. Zaki, Nermeen S. Abbas · Steroids · 2015 · 106 citations

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