Rosario Recacha

Potent, Small-Molecule Inhibitors of Human Mast Cell Tryptase. Antiasthmatic Action of a Dipeptide-Based Transition-State Analogue Containing a Benzothiazole Ketone

Michael J. Costanzo, Stephen C. Yabut, Harold R. Almond et al. · Journal of Medicinal Chemistry · 2003 · 82 citations · Full text

Life Sciences, Medicinal Chemistry, Pharmacology +14

Structural Basis for Recruitment of Rab6-Interacting Protein 1 to Golgi via a RUN Domain

Rosario Recacha, Annick Boulet, Florence Jollivet et al. · Structure · 2009 · 80 citations · Full text

Life Sciences, Cell Biology, Molecular Biology +11

Fragment-Based Discovery of 2-Aminoquinazolin-4(3<i>H</i>)-ones As Novel Class Nonpeptidomimetic Inhibitors of the Plasmepsins I, II, and IV

Dace Rasiņa, Mārtiņš Otikovs, Jānis Leitāns et al. · Journal of Medicinal Chemistry · 2015 · 65 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +16

Nonpeptide Inhibitors of Cathepsin G:  Optimization of a Novel β-Ketophosphonic Acid Lead by Structure-Based Drug Design

Michael N. Greco, Michael Hawkins, Eugene T. Powell et al. · Journal of the American Chemical Society · 2002 · 50 citations

Pharmacy, Medicinal Chemistry, Pharmacology +17

A point mutation decouples the lipid transfer activities of microsomal triglyceride transfer protein

Meredith H. Wilson, Sujith Rajan, Aidan Danoff et al. · PLoS Genetics · 2020 · 46 citations · Full text

Life Sciences, Biochemistry, Molecular Biology +17