Yann‐Vaï Le Bihan

8-Substituted Pyrido[3,4-<i>d</i>]pyrimidin-4(3<i>H</i>)-one Derivatives As Potent, Cell Permeable, KDM4 (JMJD2) and KDM5 (JARID1) Histone Lysine Demethylase Inhibitors

Vassilios Bavetsias, Rachel M. Lanigan, G.F. Ruda et al. · Journal of Medicinal Chemistry · 2016 · 97 citations · Full text

Combinatorial Chemistry, Pharmaceutical Science, Drug Target +19

The N-terminal domains of TRF1 and TRF2 regulate their ability to condense telomeric DNA

Anaïs Poulet, Sabrina Pisano, Cendrine Faivre-Moskalenko et al. · Nucleic Acids Research · 2011 · 73 citations · Full text

Genetics, Human Telomeres, Genomic Mechanism +17

Achieving <i>In Vivo</i> Target Depletion through the Discovery and Optimization of Benzimidazolone BCL6 Degraders

Benjamin R. Bellenie, Kwai-Ming J. Cheung, Ana Varela et al. · Journal of Medicinal Chemistry · 2020 · 72 citations · Full text

An Irreversible Inhibitor of HSP72 that Unexpectedly Targets Lysine‐56

Jonathan Pettinger, Yann‐Vaï Le Bihan, Marcella Widya et al. · Angewandte Chemie International Edition · 2017 · 64 citations · Full text

Bacterial Base Excision Repair Enzyme Fpg Recognizes Bulky N-Substituted-FapydG Lesion via Unproductive Binding Mode

F Coste, Matthias Ober, Yann‐Vaï Le Bihan et al. · Chemistry & Biology · 2008 · 34 citations