Kevin Shoemaker

Tests of the helix dipole model for stabilization of α-helices

Kevin Shoemaker, Peter S. Kim, Eunice J. York et al. · Nature · 1987 · 601 citations

Physics, Protein Folding, Natural Sciences +5

Identification and Characterization of NVP-BKM120, an Orally Available Pan-Class I PI3-Kinase Inhibitor

Sauveur-Michel Maira, Sabina Pecchi, Alan Huang et al. · Molecular Cancer Therapeutics · 2011 · 524 citations

Pharmacotherapy, Different Selectivity Profile, Chemical Biology +26

Discovery of Nanomolar Ligands for 7-Transmembrane G-Protein-Coupled Receptors from a Diverse N-(Substituted)glycine Peptoid Library

Ronald N. Zuckermann, Éric Martin, David C. Spellmeyer et al. · Journal of Medicinal Chemistry · 1994 · 357 citations · Full text

Nature of the charged-group effect on the stability of the C-peptide helix.

Kevin Shoemaker, Peter S. Kim, David N. Brems et al. · Proceedings of the National Academy of Sciences · 1985 · 315 citations · Full text

Identification of NVP-BKM120 as a Potent, Selective, Orally Bioavailable Class I PI3 Kinase Inhibitor for Treating Cancer

Matthew T. Burger, Sabina Pecchi, Allan S. Wagman et al. · ACS Medicinal Chemistry Letters · 2011 · 248 citations · Full text

2,4-Bismorpholino 6-Heterocyclic Pyrimidines, Pi3 Kinase Inhibitor, Orally Bioavailable Class +18