Akio Kakefuda

Nucleosides and nucleotides. 132. Synthesis and biological evaluations of ring-expanded oxetanocin analogues: Purine and pyrimidine analogues of 1,4-anhydro-2-deoxy-d-arabitol and 1,4-anhydro-2-deoxy-3-hydroxymethyl-d-arabitol

Akio Kakefuda, Satoshi Shuto, Takemitsu Nagahata et al. · Tetrahedron · 1994 · 58 citations

Natural Product Synthesis, Bioorganic Chemistry, Biochemistry +8

Welwitindolinone C synthetic studies. Construction of the welwitindolinone carbon skeleton via a transannular nitrone cycloaddition

David Freeman, A.A. Holubec, Matthew W. Weiss et al. · Tetrahedron · 2010 · 44 citations

Bioorganic Chemistry, Engineering, Heterocyclic +7

Spiro-Substituted Piperidines as Neurokinin Receptor Antagonists. III. Synthesis of (.+-.)-N-12-(3,4-Dichlorophenyl)-4-(spiro-substituted piperidin-1-yl)butyll-N-methylbenzamides and Evaluation of NK1-NK2 Dual Antagonistic Activities.

Hirokazu Kubota, Akio Kakefuda, Yoshinori Okamoto et al. · Chemical and Pharmaceutical Bulletin · 1998 · 27 citations · Full text

Spiro-substituted Piperidin-1-yl, Nk2 Receptor, Pharmacotherapy +18

Discovery of 4,5-Diphenyl-1,2,4-triazole Derivatives as a Novel Class of Selective Antagonists for the Human V1A Receptor

Akio Kakefuda · Bioorganic & Medicinal Chemistry · 2002 · 26 citations

4,5-Diphenyl-1,2,4-triazole Derivatives, Functional Selectivity, Medicine +8

Synthesis and Pharmacological Evaluation of 5-(4-Biphenyl)-3-methyl-4-phenyl-1,2,4-triazole Derivatives as a Novel Class of Selective Antagonists for the Human Vasopressin V_1A Receptor

Akio Kakefuda, Takeshi Suzuki, Takahiko Tobe et al. · Journal of Medicinal Chemistry · 2002 · 25 citations · Full text