Deheng Sun

Discovery of Potent and Noncovalent Reversible EGFR Kinase Inhibitors of EGFR^{L858R/T790M/C797S}

Qiannan Li, Tao Zhang, Shiliang Li et al. · ACS Medicinal Chemistry Letters · 2019 · 65 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +16

Novel Selective and Potent Inhibitors of Malaria Parasite Dihydroorotate Dehydrogenase: Discovery and Optimization of Dihydrothiophenone Derivatives

Minghao Xu, Junsheng Zhu, Yanyan Diao et al. · Journal of Medicinal Chemistry · 2013 · 59 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +16

Highly Selective Fluorescent Turn-On Probe for Protein Thiols in Biotin Receptor-Positive Cancer Cells

Qian Sun, Deheng Sun, Lun Song et al. · Analytical Chemistry · 2016 · 40 citations

Medicine, Biochemistry, Oncology +17

Design, Synthesis, and Biological Evaluation of Pyrimido[4,5-<i>d</i>]pyrimidine-2,4(1<i>H</i>,3<i>H</i>)-diones as Potent and Selective Epidermal Growth Factor Receptor (EGFR) Inhibitors against L858R/T790M Resistance Mutation

Yong‐Jia Hao, Jiankun Lyu, Rong Qu et al. · Journal of Medicinal Chemistry · 2018 · 37 citations · Full text

Medicine, Oncology, Pharmacology +13

Antiproliferative and apoptosis-inducing activities of novel naphthalimide–cyclam conjugates through dual topoisomerase (topo) I/II inhibition

Shaoying Tan, Deheng Sun, Jiankun Lyu et al. · Bioorganic & Medicinal Chemistry · 2015 · 31 citations

Life Sciences, Medicinal Chemistry, Pharmacology +14