Luca Carlino

Nonpeptidic Propargylamines as Inhibitors of Lysine Specific Demethylase 1 (LSD1) with Cellular Activity

Martin Schmitt, Alexander‐Thomas Hauser, Luca Carlino et al. · Journal of Medicinal Chemistry · 2013 · 75 citations · Full text

Drug Target, Pharmacotherapy, Chemical Biology +17

Synthesis, biological activity and molecular modeling studies on 1H-benzimidazole derivatives as acetylcholinesterase inhibitors

Ayşe Selcen Alpan, Sülünay Parlar, Luca Carlino et al. · Bioorganic & Medicinal Chemistry · 2013 · 67 citations · Full text

Biological Activity, 1H-benzimidazole Derivatives, Biochemistry +9

Structural basis of the effect of activating mutations on the EGF receptor

Ioannis Galdadas, Luca Carlino, Richard A. Ward et al. · eLife · 2021 · 42 citations · Full text

Molecular Biology, Cell Growth, Conformational Landscape +23

Molecular Dynamics Simulations and Classical Multidimensional Scaling Unveil New Metastable States in the Conformational Landscape of CDK2

Pasquale Pisani, Fabiana Caporuscio, Luca Carlino et al. · PLoS ONE · 2016 · 41 citations · Full text

Engineering, Biomolecular Structure Prediction, Molecular Biology +21

Structure–Activity Relationships of Hexahydrocyclopenta[<i>c</i>]quinoline Derivatives as Allosteric Inhibitors of CDK2 and EGFR

Luca Carlino, Michael S. Christodoulou, Valentina Restelli et al. · ChemMedChem · 2018 · 32 citations · Full text