Kurt A. Josef

Conformationally restrained analogs of pravadoline: nanomolar potent, enantioselective, (aminoalkyl)indole agonists of the cannabinoid receptor

Thomas E. D'Ambra, Kimberly G. Estep, Malcolm R. Bell et al. · Journal of Medicinal Chemistry · 1992 · 294 citations · Full text

Pharmacotherapy, Nanomolar Potent, Experimental Pharmacology +18

1,2-Benzothiazine 1,1-Dioxide P₂−P₃ Peptide Mimetic Aldehyde Calpain I Inhibitors

Gregory J. Wells, Ming Tao, Kurt A. Josef et al. · Journal of Medicinal Chemistry · 2001 · 163 citations · Full text

Synthesis and Structure-Activity Relationships of 6-Heterocyclic-Substituted Purines as Inactivation Modifiers of Cardiac Sodium Channels

Kimberly G. Estep, Kurt A. Josef, Edward R. Bacon et al. · Journal of Medicinal Chemistry · 1995 · 47 citations

Cardiac Muscle, Heart Failure, Inactivation Modifiers +21

Synthesis and Biological Activity of a Series of Potent Fluoromethyl Ketone Inhibitors of Recombinant Human Calpain I

Sankar Chatterjee, Mark A. Ator, Donna Bozyczko‐Coyne et al. · Journal of Medicinal Chemistry · 1997 · 45 citations

Subsite requirements for peptide aldehyde inhibitors of human calpain I

Mohamed Iqbal, Patricia A. Messina, Bethany Freed et al. · Bioorganic & Medicinal Chemistry Letters · 1997 · 44 citations

Aldo-keto Reductase, Biochemistry, Medicine +7