Concepedia
Statistics
Publications
17
Citations
567
H-Index
13
Active since
2018
Affiliations
Leipzig University(Current)
Heinrich Heine University Düsseldorf
University of Bonn
University of Tübingen
University of California San Diego
Andrea Schöler is an author at Leipzig University specializing in medicine, drug discovery, and natural sciences.
Top concepts
MedicineBiochemistryPharmacologyDrug DiscoveryNatural SciencesChemical BiologyMedicinal ChemistryDrug ResistancePharmacotherapyDrug Development
Publications per year
2018–2024
Hydroxamic Acids Immobilized on Resins (HAIRs): Synthesis of Dual‐Targeting HDAC Inhibitors and HDAC Degraders (PROTACs)
Laura Sinatra, Jan J. Bandolik, Martin Roatsch et al. · Angewandte Chemie International Edition · 2020 · 69 citations · Full text
Multicomponent Synthesis and Binding Mode of Imidazo[1,2-<i>a</i>]pyridine-Capped Selective HDAC6 Inhibitors
Marcel K. W. Mackwitz, Alexandra Hamacher, J.D. Osko et al. · Organic Letters · 2018 · 64 citations · Full text
Solid-Phase Synthesis of Cereblon-Recruiting Selective Histone Deacetylase 6 Degraders (HDAC6 PROTACs) with Antileukemic Activity
Laura Sinatra, Jing Yang, Julian Schliehe‐Diecks et al. · Journal of Medicinal Chemistry · 2022 · 63 citations · Full text
Multicomponent Synthesis, Binding Mode, and Structure–Activity Relationship of Selective Histone Deacetylase 6 (HDAC6) Inhibitors with Bifurcated Capping Groups
Nina Reßing, Melf Sönnichsen, J.D. Osko et al. · Journal of Medicinal Chemistry · 2020 · 51 citations · Full text
4-Acyl Pyrrole Capped HDAC Inhibitors: A New Scaffold for Hybrid Inhibitors of BET Proteins and Histone Deacetylases as Antileukemia Drug Leads
Linda Schäker‐Hübner, Robin Warstat, Heinz Ahlert et al. · Journal of Medicinal Chemistry · 2021 · 45 citations · Full text
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