Maarten Sijm

Lipase-Catalyzed Aza-Michael Reaction on Acrylate Derivatives

Peter Steunenberg, Maarten Sijm, Han Zuilhof et al. · The Journal of Organic Chemistry · 2013 · 43 citations

Biosynthesis, Engineering, Biochemistry +11

Targeting a Subpocket in <i>Trypanosoma brucei</i> Phosphodiesterase B1 (TbrPDEB1) Enables the Structure-Based Discovery of Selective Inhibitors with Trypanocidal Activity

Antoni R. Blaazer, Abhimanyu K. Singh, Erik de Heuvel et al. · Journal of Medicinal Chemistry · 2018 · 43 citations · Full text

Identification of the First Highly Subtype-Selective Inhibitor of Human GABA Transporter GAT3

Maria Damgaard, Anas Al-Khawaja, Stine B. Vogensen et al. · ACS Chemical Neuroscience · 2015 · 35 citations

Molecular Pharmacology, Medicinal Chemistry, Biochemistry +15

Efficacy of Novel Pyrazolone Phosphodiesterase Inhibitors in Experimental Mouse Models of Trypanosoma cruzi

Julianna Siciliano de Araújo, Cristiane França da Silva, Denise da Gama Jaén Batista et al. · Antimicrobial Agents and Chemotherapy · 2020 · 25 citations

A novel series of histamine H4 receptor antagonists based on the pyrido[3,2-d]pyrimidine scaffold: Comparison of hERG binding and target residence time with PF-3893787

Mounir Andaloussi, Herman D. Lim, Tiffany van der Meer et al. · Bioorganic & Medicinal Chemistry Letters · 2013 · 23 citations · Full text

Medicinal Chemistry, Drug Target, Novel Series +12