Concepedia

Anna Cappa

AC

6

Publications

332

Citations

6

H-Index

2014

Active since

Affiliations

European Institute of Oncology(Current)

University of Milan

University of Pavia

IFOM

Sapienza University of Rome

Anna Cappa is an author at European Institute of Oncology specializing in drug discovery, drug development, and medicine.

Top concepts

Publications per year

2014–2020

6

Publications

6

Discovery of a Novel Inhibitor of Histone Lysine-Specific Demethylase 1A (KDM1A/LSD1) as Orally Active Antitumor Agent

Paola Vianello, Oronza A. Botrugno, Anna Cappa et al. · Journal of Medicinal Chemistry · 2015 · 81 citations · Full text

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Thieno[3,2-<i>b</i>]pyrrole-5-carboxamides as New Reversible Inhibitors of Histone Lysine Demethylase KDM1A/LSD1. Part 1: High-Throughput Screening and Preliminary Exploration

Luca Sartori, Ciro Mercurio, Federica Amigoni et al. · Journal of Medicinal Chemistry · 2017 · 71 citations · Full text

Thieno[3,2-<i>b</i>]pyrrole-5-carboxamides as New Reversible Inhibitors of Histone Lysine Demethylase KDM1A/LSD1. Part 2: Structure-Based Drug Design and Structure–Activity Relationship

Paola Vianello, Luca Sartori, Federica Amigoni et al. · Journal of Medicinal Chemistry · 2017 · 70 citations · Full text

Synthesis, biological activity and mechanistic insights of 1-substituted cyclopropylamine derivatives: A novel class of irreversible inhibitors of histone demethylase KDM1A

Paola Vianello, Oronza A. Botrugno, Anna Cappa et al. · European Journal of Medicinal Chemistry · 2014 · 54 citations · Full text

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Tranylcypromine‐Based LSD1 Inhibitors: Structure‐Activity Relationships, Antiproliferative Effects in Leukemia, and Gene Target Modulation

Rossella Fioravanti, Annalisa Romanelli, Nicola Mautone et al. · ChemMedChem · 2020 · 31 citations · Full text

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