Concepedia
Statistics
Publications
32
Citations
2.9K
H-Index
25
Active since
1991
Affiliations
Pfizer (United States)(Current)
Newcastle University
Bone Therapeutics
Griffith University
Commonwealth Scientific and Industrial Research Organisation
Karen A. Maegley is an author at Pfizer (United States) specializing in medicine, drug discovery, and natural sciences.
Top concepts
MedicineBiochemistryDrug DiscoveryNatural SciencesPharmacologyMolecular BiologyDrug DevelopmentRadiation OncologyMedicinal ChemistryPharmacotherapy
Publications per year
1991–2023
Anticancer Chemosensitization and Radiosensitization by the Novel Poly(ADP-ribose) Polymerase-1 Inhibitor AG14361
Christopher Calabrese, Robert J. Almassy, Stephen Barton et al. · JNCI Journal of the National Cancer Institute · 2004 · 482 citations · Full text
Preclinical selection of a novel poly(ADP-ribose) polymerase inhibitor for clinical trial
Huw D. Thomas, Christopher Calabrese, Michael A. Batey et al. · Molecular Cancer Therapeutics · 2007 · 297 citations
Resistance-Modifying Agents. 9. Synthesis and Biological Properties of Benzimidazole Inhibitors of the DNA Repair Enzyme Poly(ADP-ribose) Polymerase
Alex W. White, Robert J. Almassy, A. Hilary Calvert et al. · Journal of Medicinal Chemistry · 2000 · 285 citations · Full text
Polycomb repressive complex 2 structure with inhibitor reveals a mechanism of activation and drug resistance
Alexei Brooun, K.S. Gajiwala, Ya‐Li Deng et al. · Nature Communications · 2016 · 158 citations · Full text
Tricyclic Benzimidazoles as Potent Poly(ADP-ribose) Polymerase-1 Inhibitors
Donald J. Skalitzky, Joseph Marakovits, Karen A. Maegley et al. · Journal of Medicinal Chemistry · 2002 · 152 citations · Full text
Medicinal Chemistry, Tricyclic Benzimidazoles, Bioorganic Chemistry +13
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