Darren Stead

Asymmetric Deprotonation of <i>N</i>-Boc Piperidine: React IR Monitoring and Mechanistic Aspects

Darren Stead, Giorgio Carbone, Peter O’Brien et al. · Journal of the American Chemical Society · 2010 · 162 citations

Asymmetric Deprotonation, Engineering, Chemical Analysis +15

Enantioselective, Palladium-Catalyzed α-Arylation of <i>N</i>-Boc Pyrrolidine: <i>In Situ</i> React IR Spectroscopic Monitoring, Scope, and Synthetic Applications

Graeme Barker, Julia L. McGrath, Artis Klapars et al. · The Journal of Organic Chemistry · 2011 · 129 citations

Engineering, Aryl Bromide, Organic Chemistry +16

Discovery of AZD9833, a Potent and Orally Bioavailable Selective Estrogen Receptor Degrader and Antagonist

James S. Scott, Amber Balazs, Bernard Barlaam et al. · Journal of Medicinal Chemistry · 2020 · 109 citations · Full text

Discovery of AZD4573, a Potent and Selective Inhibitor of CDK9 That Enables Short Duration of Target Engagement for the Treatment of Hematological Malignancies

Bernard Barlaam, Robert Casella, Justin Cidado et al. · Journal of Medicinal Chemistry · 2020 · 98 citations · Full text

Isothiourea-Catalyzed Enantioselective Addition of 4-Nitrophenyl Esters to Iminium Ions

Jude N. Arokianathar, Aileen B. Frost, Alexandra M. Z. Slawin et al. · ACS Catalysis · 2017 · 70 citations · Full text