Daniel Conole

3,5-Dialkoxypyridine analogues of bedaquiline are potent antituberculosis agents with minimal inhibition of the hERG channel

Hamish S. Sutherland, Amy S.T. Tong, Peter J. Choi et al. · Bioorganic & Medicinal Chemistry · 2019 · 109 citations · Full text

Pharmaceutical Science, 3,5-Dialkoxypyridine Analogues, Herg Channel +20

6-Cyano Analogues of Bedaquiline as Less Lipophilic and Potentially Safer Diarylquinolines for Tuberculosis

Amy S.T. Tong, Peter J. Choi, Adrian Blaser et al. · ACS Medicinal Chemistry Letters · 2017 · 79 citations · Full text

Structure-activity relationships for analogs of the tuberculosis drug bedaquiline with the naphthalene unit replaced by bicyclic heterocycles

Hamish S. Sutherland, Amy S.T. Tong, Peter J. Choi et al. · Bioorganic & Medicinal Chemistry · 2018 · 76 citations · Full text

Riociguat: First Global Approval

Daniel Conole, Lesley J. Scott · Drugs · 2013 · 61 citations

International Research, Humanities, First Global Approval +9

Structure-activity relationships for unit C pyridyl analogues of the tuberculosis drug bedaquiline

Adrian Blaser, Hamish S. Sutherland, Amy S.T. Tong et al. · Bioorganic & Medicinal Chemistry · 2019 · 51 citations · Full text