Adrian Blaser

5-Substituted 2-Aminopyridine <i>C</i>-Nucleosides as Protonated Cytidine Equivalents:  Increasing Efficiency and Selectivity in DNA Triple-Helix Formation

Stefan Hildbrand, Adrian Blaser, Serge P. Parel et al. · Journal of the American Chemical Society · 1997 · 113 citations

Life Sciences, Biochemistry, Molecular Biology +17

Synthesis and Structure–Activity Relationships of Varied Ether Linker Analogues of the Antitubercular Drug (6<i>S</i>)-2-Nitro-6-{[4-(trifluoromethoxy)benzyl]oxy}-6,7-dihydro-5<i>H</i>-imidazo[2,1-<i>b</i>][1,3]oxazine (PA-824)

Andrew M. Thompson, Hamish S. Sutherland, Brian D. Palmer et al. · Journal of Medicinal Chemistry · 2011 · 109 citations

Pharmacy, Medicinal Chemistry, Pharmacology +16

Synthesis and Structure−Activity Studies of Biphenyl Analogues of the Tuberculosis Drug (6<i>S</i>)-2-Nitro-6-{[4-(trifluoromethoxy)benzyl]oxy}-6,7-dihydro-5<i>H</i>-imidazo[2,1-<i>b</i>][1,3]oxazine (PA-824)

Brian D. Palmer, Andrew M. Thompson, Hamish S. Sutherland et al. · Journal of Medicinal Chemistry · 2009 · 109 citations · Full text

Pharmacy, Chemistry, Medicinal Chemistry +11

Synthesis, Reduction Potentials, and Antitubercular Activity of Ring A/B Analogues of the Bioreductive Drug (6<i>S</i>)-2-Nitro-6-{[4-(trifluoromethoxy)benzyl]oxy}-6,7-dihydro-5<i>H</i>-imidazo[2,1-<i>b</i>][1,3]oxazine (PA-824)

Andrew M. Thompson, Adrian Blaser, Robert F. Anderson et al. · Journal of Medicinal Chemistry · 2008 · 93 citations

Pharmacy, Medicinal Chemistry, Pharmacology +12

Synthesis and Structure−activity Relationships of Antitubercular 2-Nitroimidazooxazines Bearing Heterocyclic Side Chains

Hamish S. Sutherland, Adrian Blaser, Iveta Kmentová et al. · Journal of Medicinal Chemistry · 2009 · 89 citations

Pharmacy, Medicinal Chemistry, Pharmacology +13