Westley Tear

Progress against <i>Escherichia coli</i> with the Oxazolidinone Class of Antibacterials: Test Case for a General Approach To Improving Whole-Cell Gram-Negative Activity

Khuloud Takrouri, Harold D. Cooper, Andrew Spaulding et al. · ACS Infectious Diseases · 2016 · 31 citations

Hybrid C-ring Analogues, Bioorganic Chemistry, Escherichia Coli +24

From Cells to Mice to Target: Characterization of NEU-1053 (SB-443342) and Its Analogues for Treatment of Human African Trypanosomiasis

William G. Devine, Rosario Díaz-González, Gloria Ceballos-Pérez et al. · ACS Infectious Diseases · 2017 · 21 citations · Full text

Selectivity and Physicochemical Optimization of Repurposed Pyrazolo[1,5-<i>b</i>]pyridazines for the Treatment of Human African Trypanosomiasis

Westley Tear, Seema Bag, Rosario Díaz-González et al. · Journal of Medicinal Chemistry · 2019 · 17 citations · Full text

Compound design guidelines for evading the efflux and permeation barriers of Escherichia coli with the oxazolidinone class of antibacterials: Test case for a general approach to improving whole cell Gram-negative activity

Andrew Spaulding, Khuloud Takrouri, Pornachandran Mahalingam et al. · Bioorganic & Medicinal Chemistry Letters · 2017 · 16 citations

Antimicrobial Susceptibility, Antibiotics, Medicine +10

Discovery and SAR Study of Boronic Acid-Based Selective PDE3B Inhibitors from a Novel DNA-Encoded Library

Ann Rowley, Gang Yao, Logan D. Andrews et al. · Journal of Medicinal Chemistry · 2024 · 10 citations