Marek Cebrat

Structure of the GCN5 histone acetyltransferase bound to a bisubstrate inhibitor

A.N. Poux, Marek Cebrat, Cheol M. Kim et al. · Proceedings of the National Academy of Sciences · 2002 · 109 citations · Full text

Crystal Structure, Molecular Biology, Chemical Biology +17

Histone Acetyltransferase Activity of p300 Is Required for Transcriptional Repression by the Promyelocytic Leukemia Zinc Finger Protein

Fabien Guidez, Louise Howell, Mark Isalan et al. · Molecular and Cellular Biology · 2005 · 105 citations · Full text

Histone Modifications, Epigenetic Change, Molecular Biology +16

Synthesis and analysis of potential prodrugs of coenzyme A analogues for the inhibition of the histone acetyltransferase p300

Marek Cebrat, Cheol M. Kim, Paul R. Thompson et al. · Bioorganic & Medicinal Chemistry · 2003 · 71 citations

Potential Prodrugs, Medicinal Chemistry, Biosynthesis +13

Synthesis and Evaluation of a Potent and Selective Cell-Permeable p300 Histone Acetyltransferase Inhibitor

Y. George Zheng, Karanam Balasubramanyam, Marek Cebrat et al. · Journal of the American Chemical Society · 2005 · 68 citations

Medicinal Chemistry, P300-sensitive Reporter, Signal Transduction +12

p300/CBP-associated Factor Drives DEK into Interchromatin Granule Clusters

Joanne Cleary, Kajal Sitwala, Michael S. Khodadoust et al. · Journal of Biological Chemistry · 2005 · 65 citations · Full text

Chromatin, Chromatin Structure, Chromatin Remodeling +14