Judith Borsboom

Discovery of selective and orally available spiro-3-piperidyl ATP-competitive MK2 inhibitors

Allard Kaptein, Arthur Oubrie, Edwin de Zwart et al. · Bioorganic & Medicinal Chemistry Letters · 2011 · 19 citations · Full text

Medicinal Chemistry, Biochemistry, Medicine +9

Asymmetric Synthesis of (<i>S</i>)‐Mirtazapine: Unexpected Racemization through an Aromatic <i>ipso</i>‐Attack Mechanism

Marco van der Linden, Judith Borsboom, Frans M. Kaspersen et al. · European Journal of Organic Chemistry · 2008 · 15 citations

Diversity Oriented Synthesis, Natural Product Synthesis, Engineering +13

Novel ATP competitive MK2 inhibitors with potent biochemical and cell-based activity throughout the series

Arthur Oubrie, Allard Kaptein, Edwin de Zwart et al. · Bioorganic & Medicinal Chemistry Letters · 2011 · 14 citations · Full text

Cell-based Activity, Novel Therapy, Biochemistry +8