Killian Oukoloff - Concepedia

Author

Killian Oukoloff

University of California San Diego

Also Known As

Killian Oukoloff, Oukoloff, Killian

Publications

510

Citations

H-Index

Concepts

All Affiliations

University of California San Diego University of Pennsylvania University of Montana Laboratoire COBRA Normandie Université

About

Killian Oukoloff is an author at University of California San Diego specializing in biochemistry, medicine, and pharmacology.

Top Concepts

#	Concept	H-Index	Publications	Citations
1	Medicine	3	3	139
2	Natural Sciences	3	3	167
3	Biochemistry	3	3	167
4	Biomolecular Engineering	1	1	48
5	Chemistry	1	1	26

Killian Oukoloff

Publications

358

Citations

H-Index

Page 1

	Year	Citations
Design, biological evaluation and X-ray crystallography of nanomolar multifunctional ligands targeting simultaneously acetylcholinesterase and glycogen synthase kinase-3 Killian Oukoloff, Nicolas Coquelle, Manuela Bartolini, European Journal of Medicinal Chemistry X-ray CrystallographyProtein AssemblyBiochemistryNanomolar Multifunctional LigandsNatural Sciences	2019	65
Evaluation of Oxetan-3-ol, Thietan-3-ol, and Derivatives Thereof as Bioisosteres of the Carboxylic Acid Functional Group Pierrik Lassalas, Killian Oukoloff, Vishruti Makani, ACS Medicinal Chemistry Letters Medicinal ChemistryEnantioselective SynthesisBioorganic ChemistryDerivativesBiochemistry	2017	54
Multitargeted Imidazoles: Potential Therapeutic Leads for Alzheimer’s and Other Neurodegenerative Diseases Anne‐Sophie Cornec, Ludovica Monti, Jane Kovalevich, Journal of Medicinal Chemistry Drug Target5-Lox-derived EicosanoidsNeurochemical BiomarkersPharmacotherapyPharmaceutical Chemistry	2017	48
A brain-penetrant triazolopyrimidine enhances microtubule-stability, reduces axonal dysfunction and decreases tau pathology in a mouse tauopathy model Bin Zhang, Yuemang Yao, Anne‐Sophie Cornec, Molecular Neurodegeneration	2018	41
Evaluation of the Structure–Activity Relationship of Microtubule-Targeting 1,2,4-Triazolo[1,5-<i>a</i>]pyrimidines Identifies New Candidates for Neurodegenerative Tauopathies Killian Oukoloff, Goodwell Nzou, Carmine Varricchio, Journal of Medicinal Chemistry	2021	28
Brain‐Penetrant Triazolopyrimidine and Phenylpyrimidine Microtubule Stabilizers as Potential Leads to Treat Human African Trypanosomiasis Ludovica Monti, Steven C Wang, Killian Oukoloff, ChemMedChem	2018	27
Design, synthesis and evaluation of photoactivatable derivatives of microtubule (MT)-active [1,2,4]triazolo[1,5-a]pyrimidines Killian Oukoloff, Jane Kovalevich, Anne‐Sophie Cornec, Bioorganic & Medicinal Chemistry Letters Photoactivatable DerivativesDerivative (Chemistry)DerivativesPhotochemistryMedicine	2018	26
Microtubule-Stabilizing 1,2,4-Triazolo[1,5-<i>a</i>]pyrimidines as Candidate Therapeutics for Neurodegenerative Disease: Matched Molecular Pair Analyses and Computational Studies Reveal New Structure–Activity Insights Thibault Alle, Carmine Varricchio, Yuemang Yao, Journal of Medicinal Chemistry	2022	17
Inhibition of the HEG1–KRIT1 interaction increases KLF4 and KLF2 expression in endothelial cells Miguel Alejandro Lopez‐Ramirez, Sara McCurdy, Wenqing Li, FASEB BioAdvances	2021	16
Discovery, Optimization, and Preclinical Pharmacology of EP652, a METTL3 Inhibitor with Efficacy in Liquid and Solid Tumor Models Guillaume Dutheuil, Killian Oukoloff, Julien Korac, Journal of Medicinal Chemistry	2025	14

Page 1