Tom McInally

Hit-to-Lead studies: The discovery of potent adamantane amide P2X7 receptor antagonists

Andrew Baxter, Janice Bent, Keith Bowers et al. · Bioorganic & Medicinal Chemistry Letters · 2003 · 117 citations · Full text

Drug Target, Biochemistry, Functional Selectivity +9

1,2-Dihydro-4-quinazolinamines:  Potent, Highly Selective Inhibitors of Inducible Nitric Oxide Synthase Which Show Antiinflammatory Activity in Vivo

Alan C. Tinker, Haydn G. Beaton, N. K. Boughton-Smith et al. · Journal of Medicinal Chemistry · 2003 · 95 citations · Full text

Highly Selective Inhibitors, Medicinal Chemistry, Bioorganic Chemistry +15

Hit-to-lead studies: the discovery of potent, orally active, thiophenecarboxamide IKK-2 inhibitors

Andrew Baxter, Steve Brough, Anne Cooper et al. · Bioorganic & Medicinal Chemistry Letters · 2004 · 90 citations

Medicinal Chemistry, Thiophenecarboxamide Ikk-2 Inhibitors, Hit Identification +11

Acyl radical cyclisation onto pyrroles

Steven M. Allin, William Barton, W. Russell Bowman et al. · Tetrahedron Letters · 2001 · 69 citations

Heterocyclic, Radical (Chemistry), Acyl Radical Cyclisation +3

Radical cyclisation onto pyrazoles: synthesis of withasomnine

Steven M. Allin, William Barton, W. Russell Bowman et al. · Tetrahedron Letters · 2002 · 57 citations

Radical Cyclisation, Organic Chemistry, Heterocycle Chemistry +2