Michael L. Denney

Dibasic Benzo[<i>b</i>]thiophene Derivatives as a Novel Class of Active Site-Directed Thrombin Inhibitors. 1. Determination of the Serine Protease Selectivity, Structure−Activity Relationships, and Binding Orientation

Daniel J. Sall, Jolie Bastian, John A. Buben et al. · Journal of Medicinal Chemistry · 1997 · 54 citations

Pharmacy, Medicinal Chemistry, Pharmacology +10

Dibasic benzo[b]thiophene derivatives as a novel class of active site directed thrombin inhibitors: 4. SAR studies on the conformationally restricted C3-side chain of hydroxybenzo[b]thiophenes

Kumiko Takeuchi, Todd J. Kohn, Daniel J. Sall et al. · Bioorganic & Medicinal Chemistry Letters · 1999 · 35 citations

Pharmacy, Chemistry, Medicinal Chemistry +12

Diamino Benzo[<i>b</i>]thiophene Derivatives as a Novel Class of Active Site Directed Thrombin Inhibitors. 5. Potency, Efficacy, and Pharmacokinetic Properties of Modified C-3 Side Chain Derivatives

Daniel J. Sall, Dianna L. Bailey, Jolie Bastian et al. · Journal of Medicinal Chemistry · 2000 · 31 citations

Pharmacy, Medicinal Chemistry, Pharmacology +17

Use of Conformationally Restricted Benzamidines as Arginine Surrogates in the Design of Platelet GPIIb-IIIa Receptor Antagonists

Daniel J. Sall, Ann Arfsten, Jolie Bastian et al. · Journal of Medicinal Chemistry · 1997 · 22 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Dibasic benzo[b]thiophene derivatives as a novel class of active site directed thrombin inhibitors: 2: sidechain optimization and demonstration of in vivo efficacy

Minsheng Zhang, Dianna L. Bailey, Jolie Bastian et al. · Bioorganic & Medicinal Chemistry Letters · 1999 · 13 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +11