Concepedia

Christian L. Holst

CL

Statistics

Publications

5

Citations

110

H-Index

5

Active since

2002

Affiliations

Albany Molecular Research (United States)(Current)

Bristol-Myers Squibb (United States)

Bristol-Myers Squibb (Germany)

Bristol-Myers Squibb (Sweden)

Christian L. Holst is an author at Albany Molecular Research (United States) specializing in medicinal chemistry, pharmacy, and pharmacology.

Publications per year

2002–2016

5

Publications

5

Discovery and Preclinical Evaluation of [4-[[1-(3-fluorophenyl)methyl]-1<i>H</i>-indazol-5-ylamino]-5-methylpyrrolo[2,1-<i>f</i>][1,2,4]triazin-6-yl]carbamic Acid, (3<i>S</i>)-3-Morpholinylmethyl Ester (BMS-599626), a Selective and Orally Efficacious Inhibitor of Human Epidermal Growth Factor Receptor 1 and 2 Kinases

Ashvinikumar V. Gavai, Brian E. Fink, David J. Fairfax et al. · Journal of Medicinal Chemistry · 2009 · 30 citations · Full text

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Discovery of silyl proline containing HCV NS5A inhibitors with pan-genotype activity: SAR development

Anilkumar G. Nair, Qingbei Zeng, Oleg Selyutin et al. · Bioorganic & Medicinal Chemistry Letters · 2016 · 27 citations · Full text

, , +15

Total Synthesis of Gibbilimbols A−D

James R. Vyvyan, Christian L. Holst, Allison J. Johnson et al. · The Journal of Organic Chemistry · 2002 · 22 citations

, , +12

Discovery of BMS-641988, a Novel Androgen Receptor Antagonist for the Treatment of Prostate Cancer

Aaron Balog, Richard Rampulla, Greg S. Martin et al. · ACS Medicinal Chemistry Letters · 2015 · 20 citations · Full text

, , +17

Design and synthesis of 4-[3,5-dioxo-11-oxa-4,9-diazatricyclo[5.3.1.02,6]undec-4-yl]-2-trifluoromethyl-benzonitriles as androgen receptor antagonists

Hai‐Yun Xiao, Aaron Balog, Ricardo M. Attar et al. · Bioorganic & Medicinal Chemistry Letters · 2010 · 11 citations · Full text

, , +10

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