Marian V. Gorichko

Open science discovery of potent noncovalent SARS-CoV-2 main protease inhibitors

Melissa L. Boby, D. Fearon, Matteo P. Ferla et al. · Science · 2023 · 158 citations · Full text

Synthesis of 3-heteryl substituted pyrrolidine-2,5-diones via catalytic Michael reaction and evaluation of their inhibitory activity against InhA and Mycobacterium tuberculosis

Tetiana Matviiuk, Giorgia Mori, Christian Lherbet et al. · European Journal of Medicinal Chemistry · 2013 · 49 citations

Inhibitory Activity, Engineering, Heterocyclic +6

Design, chemical synthesis of 3-(9H-fluoren-9-yl)pyrrolidine-2,5-dione derivatives and biological activity against enoyl-ACP reductase (InhA) and Mycobacterium tuberculosis

Tetiana Matviiuk, Frédéric Rodriguez, N. Saffon et al. · European Journal of Medicinal Chemistry · 2013 · 45 citations

Biochemistry, Enoyl-acp Reductase, Medicine +7

Turning high-throughput structural biology into predictive inhibitor design

Kadi L. Saar, William McCorkindale, D. Fearon et al. · Proceedings of the National Academy of Sciences · 2023 · 22 citations · Full text

Hetaryl Bromides Bearing the SO₂F Group – Versatile Substrates for Palladium‐Catalyzed C–C Coupling Reactions

Artem Cherepakha, Kateryna O. Stepannikova, Bohdan V. Vashchenko et al. · European Journal of Organic Chemistry · 2018 · 21 citations

Chemical Engineering, Cross-coupling Reaction, Derivatives +14