Concepedia

Frédéric Labéguère

FL

Statistics

Publications

4

Citations

158

H-Index

4

Active since

2002

Affiliations

Galapagos (France)(Current)

Galapagos (Belgium)

University of Glasgow

Frédéric Labéguère is an author at Galapagos (France) specializing in ligand binding, molecular pharmacology, and medicinal chemistry.

Publications per year

2002–2023

4

Publications

4

Three classes of ligands each bind to distinct sites on the orphan G protein-coupled receptor GPR84

Zobaer Al Mahmud, Laura Jenkins, Trond Ulven et al. · Scientific Reports · 2017 · 49 citations · Full text

, , +17

Discovery of 9-Cyclopropylethynyl-2-((<i>S</i>)-1-[1,4]dioxan-2-ylmethoxy)-6,7-dihydropyrimido[6,1-<i>a</i>]isoquinolin-4-one (GLPG1205), a Unique GPR84 Negative Allosteric Modulator Undergoing Evaluation in a Phase II Clinical Trial

Frédéric Labéguère, Sonia Dupont, Luke J. Alvey et al. · Journal of Medicinal Chemistry · 2020 · 46 citations · Full text

, , +17

IRAK4 inhibition dampens pathogenic processes driving inflammatory skin diseases

Stéphanie Lavazais, Manja Jargosch, Sonia Dupont et al. · Science Translational Medicine · 2023 · 40 citations

, , +17

An efficient diastereoselective synthesis of β-1-formyl-2,3,4,6-tetra-O-benzyl-d-glucopyranoside

Frédéric Labéguère, Jean‐Pierre Lavergne, Jean Martínez · Tetrahedron Letters · 2002 · 23 citations

, , +8

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