Concepedia
5
Publications
168
Citations
H-Index
2019
Active since
Affiliations
Takeda (Japan)(Current)
Swiss Tropical and Public Health Institute
WuXi AppTec (China)
Eisai (Japan)
Griffith University
Yuichiro Akao is an author at Takeda (Japan).
Publications per year
2019–2024
Optimization of Methionyl tRNA-Synthetase Inhibitors for Treatment of <i>Cryptosporidium</i> Infection
Frederick S. Buckner, Ranae M. Ranade, J. Robert Gillespie et al. · Antimicrobial Agents and Chemotherapy · 2019 · 50 citations · Full text
Collaborative virtual screening to elaborate an imidazo[1,2- <i>a</i> ]pyridine hit series for visceral leishmaniasis
Yuichiro Akao, Stacie Canan, Yafeng Cao et al. · RSC Medicinal Chemistry · 2021 · 39 citations · Full text
Discovery and Structure–Activity Relationships of Quinazolinone-2-carboxamide Derivatives as Novel Orally Efficacious Antimalarials
Benoı̂t Laleu, Yuichiro Akao, Atsuko Ochida et al. · Journal of Medicinal Chemistry · 2021 · 35 citations · Full text
Repositioning and Characterization of 1-(Pyridin-4-yl)pyrrolidin-2-one Derivatives as <i>Plasmodium</i> Cytoplasmic Prolyl-tRNA Synthetase Inhibitors
Masanori Okaniwa, Akira Shibata, Atsuko Ochida et al. · ACS Infectious Diseases · 2021 · 25 citations · Full text
High-throughput screening of small-molecules libraries identified antibacterials against clinically relevant multidrug-resistant A. baumannii and K. pneumoniae
Benjamin Blasco, Soojin Jang, Hiroki Terauchi et al. · EBioMedicine · 2024 · 19 citations · Full text
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