Heather Coate

Novel 2-phenylquinolin-7-yl-derived imidazo[1,5-a]pyrazines as potent insulin-like growth factor-I receptor (IGF-IR) inhibitors

Mark J. Mulvihill, Qunsheng Ji, Heather Coate et al. · Bioorganic & Medicinal Chemistry · 2007 · 72 citations · Full text

Medicinal Chemistry, Biochemistry, Medicine +9

GPR139, an Orphan Receptor Highly Enriched in the Habenula and Septum, Is Activated by the Essential Amino Acids l-Tryptophan and l-Phenylalanine

Changlu Liu, Pascal Bonaventure, Grace Lee et al. · Molecular Pharmacology · 2015 · 72 citations

Pharmacological Blockade of the DP2 Receptor Inhibits Cigarette Smoke-Induced Inflammation, Mucus Cell Metaplasia, and Epithelial Hyperplasia in the Mouse Lung

Karin J. Stebbins, Alex Broadhead, Christopher Baccei et al. · Journal of Pharmacology and Experimental Therapeutics · 2009 · 48 citations

Novel tricyclic antagonists of the prostaglandin D2 receptor DP2 with efficacy in a murine model of allergic rhinitis

Brian A. Stearns, Christopher Baccei, Gretchen Bain et al. · Bioorganic & Medicinal Chemistry Letters · 2009 · 45 citations · Full text

Inflammation, Allergy, Allergy Medicine +10

Amino substituted analogs of 1-phenyl-3-phenylimino-2-indolones with potent galanin Gal3 receptor binding affinity and improved solubility

Michael J. Konkel, Mathivanan Packiarajan, Heidi Chen et al. · Bioorganic & Medicinal Chemistry Letters · 2006 · 37 citations · Full text

Medicinal Chemistry, Bioorganic Chemistry, Biochemistry +7