Christian K. Sams

Optimization of Alkylidene Hydrazide Based Human Glucagon Receptor Antagonists. Discovery of the Highly Potent and Orally Available 3-Cyano-4-hydroxybenzoic Acid [1-(2,3,5,6-Tetramethylbenzyl)-1<i>H</i>-indol-4-ylmethylene]hydrazide

Peter Madsen, Anthony Ling, Michael Plewe et al. · Journal of Medicinal Chemistry · 2002 · 87 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

New β-Alanine Derivatives Are Orally Available Glucagon Receptor Antagonists

Jesper Lau, Carsten Behrens, Ulla G. Sidelmann et al. · Journal of Medicinal Chemistry · 2007 · 53 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +16

Novel Glucagon Receptor Antagonists with Improved Selectivity over the Glucose-Dependent Insulinotropic Polypeptide Receptor

János T. Kodra, Anker Jørgensen, Birgitte Andersen et al. · Journal of Medicinal Chemistry · 2008 · 53 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +16

Human glucagon receptor antagonists based on alkylidene hydrazides

Anthony Ling, Michael Plewe, Javier González et al. · Bioorganic & Medicinal Chemistry Letters · 2002 · 40 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +14

Solid-phase synthesis of 1,2,4-oxadiazoles

Christian K. Sams, Jesper Lau · Tetrahedron Letters · 1999 · 17 citations

Natural Sciences, Chemistry, Solid-state Chemistry +5