René Trussardi

Industrial Synthesis of the Key Precursor in the Synthesis of the Anti-Influenza Drug Oseltamivir Phosphate (Ro 64-0796/002, GS-4104-02):  Ethyl (3<i>R</i>,4<i>S</i>,5<i>S</i>)-4,5-epoxy-3-(1-ethyl-propoxy)-cyclohex-1-ene-1-carboxylate

Muriel Federspiel, R. Fischer, Michael Hennig et al. · Organic Process Research & Development · 1999 · 155 citations

Pharmacy, Chemistry, Medicinal Chemistry +8

New, Azide-Free Transformation of Epoxides into 1,2-Diamino Compounds:  Synthesis of the Anti-Influenza Neuraminidase Inhibitor Oseltamivir Phosphate (Tamiflu)

Martin Karpf, René Trussardi · The Journal of Organic Chemistry · 2001 · 140 citations

Pharmacy, Medicinal Chemistry, Pharmacology +15

The Synthetic Development of the Anti-Influenza Neuraminidase Inhibitor Oseltamivir Phosphate (Tamiflu®): A Challenge for Synthesis &amp; Process Research

Stefan Abrecht, Peter J. Harrington, Hans Iding et al. · CHIMIA International Journal for Chemistry · 2004 · 130 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +13

Efficient Access to Oseltamivir Phosphate (Tamiflu) via the <i>O‐</i>Trimesylate of Shikimic Acid Ethyl Ester

Martin Karpf, René Trussardi · Angewandte Chemie International Edition · 2009 · 80 citations

Pharmacy, Medicinal Chemistry, Pharmacology +7