B. Garnham

Regioselective structural and functional mimicry of peptides. Design of hydrolytically-stable cyclic peptidomimetic inhibitors of HIV-1 protease.

Giovanni Abbenante, Darren R. March, Douglas A. Bergman et al. · Journal of the American Chemical Society · 1995 · 58 citations

Peptide Engineering, Altmetric Attention Score, Peptide Science +16

A novel thioether linker: Chemical synthesis of a HIV-1 protease analogue by thioether ligation

Darren R. Englebretsen, B. Garnham, Douglas A. Bergman et al. · Tetrahedron Letters · 1995 · 54 citations

Medicinal Chemistry, Bioorganic Chemistry, Biochemistry +9

Solid phase synthesis of hydroxyethylamine peptide bond isosteres: Synthesis of the potent HIV-1 protease inhibitor JG365

Paul F. Alewood, Ross I. Brinkworth, Robert J. Dancer et al. · Tetrahedron Letters · 1992 · 25 citations

Medicinal Chemistry, Biochemistry, Natural Sciences +9

Structure-activity relationships for macrocyclic peptidomimetic inhibitors of HIV-1 protease

Giovanni Abbenante, Douglas A. Bergman, R.I. Brinkworth et al. · Bioorganic & Medicinal Chemistry Letters · 1996 · 14 citations

Hiv-1 Protease, Medicine, Peptoid +4

A Cassette Ligation Strategy with Thioether Replacement of Three Gly-Gly Peptide Bonds: Total Chemical Synthesis of the 101 Residue Protein Early Pregnancy Factor [ψ(CH₂S)²⁸^-^29,56^-^57,76^-⁷⁷]

Darren R. Englebretsen, B. Garnham, Paul F. Alewood · The Journal of Organic Chemistry · 2002 · 13 citations