Songfeng Lu

<i>N</i>-(Cycloalkylamino)acyl-2-aminothiazole Inhibitors of Cyclin-Dependent Kinase 2. <i>N</i>-[5-[[[5-(1,1-Dimethylethyl)-2-oxazolyl]methyl]thio]-2-thiazolyl]-4- piperidinecarboxamide (BMS-387032), a Highly Efficacious and Selective Antitumor Agent

Raj N. Misra, Hai‐Yun Xiao, Kyoung S. Kim et al. · Journal of Medicinal Chemistry · 2004 · 251 citations · Full text

Chemoprevention Strategy, Immunology, Pharmacotherapy +19

Discovery of Aminothiazole Inhibitors of Cyclin-Dependent Kinase 2:  Synthesis, X-ray Crystallographic Analysis, and Biological Activities

Kyoung Soon Kim, S. David Kimball, Raj N. Misra et al. · Journal of Medicinal Chemistry · 2002 · 156 citations · Full text

Combinatorial Chemistry, Drug Target, Cdk2 Protein +20

Synthesis and Biological Evaluation of 3-Aryl-3-(4-phenoxy)-propionic Acid as a Novel Series of G Protein-Coupled Receptor 40 Agonists

Fengbin Song, Songfeng Lu, Joe Gunnet et al. · Journal of Medicinal Chemistry · 2007 · 91 citations · Full text

Pharmacotherapy, Insulin Signaling, Metabolic Syndrome +20

Probing the bradykinin receptor: mapping the geometric topography using ethers of hydroxyproline in novel peptides

Donald J. Kyle, Jennifer A. Martin, Ronald M. Burch et al. · Journal of Medicinal Chemistry · 1991 · 68 citations

Peptide Engineering, Peptide Science, System Pharmacology +19

Synthesis and biological activity of N-aryl-2-aminothiazoles: potent pan inhibitors of cyclin-dependent kinases

Raj N. Misra, Hai‐Yun Xiao, David Williams et al. · Bioorganic & Medicinal Chemistry Letters · 2004 · 56 citations · Full text

Biological Activity, Cyclin-dependent Kinases, Biochemistry +10