Discovery of a potent and selective small molecule hGPR91 antagonist

Debnath Bhuniya, Dhananjay N. Umrani, Bhavesh Dave, +24

Bioorganic & Medicinal Chemistry Letters

Drug TargetFunctional SelectivityMedicineG Protein-coupled ReceptorReceptor (Biochemistry) +6

Modulation of Dopamine Receptor Agonist-Induced Rotational Behavior in 6-OHDA-Lesioned Rats by a Peptidomimetic Analogue of Pro-Leu-Gly-NH2 (PLG)

Ram K. Mishra, Éric Marcotte, Anita Chugh, +3

Peptides

Peptidomimetic AnalogueFunctional SelectivityMedicinePhysiologyNeuropeptide Receptor +8

Endothelin-receptor antagonists: current and future perspectives

Abhijit Ray, Laxminarayan G. Hegde, Anita Chugh, +1

Drug Discovery Today

Molecular PhysiologyMedicinePhysiologyEndothelial DysfunctionVascular Biology +3

Design and synthesis of novel xanthine derivatives as potent and selective A 2B adenosine receptor antagonists for the treatment of chronic inflammatory airway diseases

Sujay Basu, Dinesh A. Barawkar, Ramdas Vidya, +24

European Journal of Medicinal Chemistry

AsthmaMedicinal ChemistryAnti-inflammatoryAllergyInflammatory Lung Disease +8

Protection Against MPTP Treatment by an Analog of Pro-Leu-Gly-NH2 (PLG, MIF-1)

Éric Marcotte, Anita Chugh, Ram K. Mishra, +1

Peptides

PharmacologyMolecular PharmacologyMedicineBiochemistry

A 2B adenosine receptor antagonists: Design, synthesis and biological evaluation of novel xanthine derivatives

Sujay Basu, Dinesh A. Barawkar, Ramdas Vidya, +26

European Journal of Medicinal Chemistry

BiochemistryFunctional SelectivityMedicineNovel Xanthine DerivativesMechanism Of Action +6

Opposing effect of apomorphine on antinociceptive activityfx of morphine: a dose-dependent phenomenon

Yogendra Kumar Gupta, Anita Chugh, Shikha Seth

Pain

Potent and Selective Inhibitors of Long Chain <scp>l</scp>-2-Hydroxy Acid Oxidase Reduced Blood Pressure in DOCA Salt-Treated Rats

Dinesh A. Barawkar, Ashwin Meru, Anish Bandyopadhyay, +28

ACS Medicinal Chemistry Letters

Molecular PharmacologyHypertensionBiochemistrySelective Hao2 InhibitorsMedicine +12

Role of peripheral 5-HT1A receptors in detrusor over activity associated with partial bladder outlet obstruction in female rats

Shivani Mittra, Shivani Malhotra, Krishna S. Naruganahalli, +1

European Journal of Pharmacology

Urological ResearchUrologyVoiding DysfunctionMedicineHormonal Receptor +7

Discovery of liver-directed glucokinase activator having anti-hyperglycemic effect without hypoglycemia

Anil M. Deshpande, Debnath Bhuniya, Siddhartha De, +22

European Journal of Medicinal Chemistry

Metabolic SyndromeDiabetes ManagementBiochemistryMedicineLiver Physiology +9