Arkadii Vaisburg

Novel Aminophenyl Benzamide-Type Histone Deacetylase Inhibitors with Enhanced Potency and Selectivity

Oscar Moradei, Tammy C. Mallais, Sylvie Fréchette et al. · Journal of Medicinal Chemistry · 2007 · 164 citations · Full text

Pharmacy, Medicinal Chemistry, Oncology +16

Discovery of <i>N</i>-(2-Aminophenyl)-4-[(4-pyridin-3-ylpyrimidin-2-ylamino)methyl]benzamide (MGCD0103), an Orally Active Histone Deacetylase Inhibitor

Nancy Zhou, Oscar Moradei, Stéphane Raeppel et al. · Journal of Medicinal Chemistry · 2008 · 108 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +13

Structurally Simple Trichostatin A-Like Straight Chain Hydroxamates as Potent Histone Deacetylase Inhibitors

Soon Hyung Woo, Sylvie Fréchette, Elie Abou Khalil et al. · Journal of Medicinal Chemistry · 2002 · 72 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +14

Discovery of a novel and potent series of thieno[3,2-b]pyridine-based inhibitors of c-Met and VEGFR2 tyrosine kinases

Stephen Claridge, Franck Raeppel, Marie‐Claude Granger et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 63 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +13

Metabolic targeting of cancer by a ubiquinone uncompetitive inhibitor of mitochondrial complex I

Shashi Jain, Cheng Hu, Jérôme Kluza et al. · Cell chemical biology · 2021 · 60 citations

Life Sciences, Oncology, Pharmacology +14