Graham L. Simpson - Concepedia

Author

Graham L. Simpson

GlaxoSmithKline (United Kingdom)

Also Known As

G. Simpson, Graham L Simpson, Graham L. Simpson, Graham L. Simpson (1523503), Graham Simpson

Publications

692

Citations

H-Index

Concepts

All Affiliations

GlaxoSmithKline (United Kingdom)Massachusetts Institute of Technology GlaxoSmithKline (United States)South College University of Glasgow

About

Graham L. Simpson is an author at GlaxoSmithKline (United Kingdom) specializing in medicine, natural sciences, and molecular biology.

Top Concepts

#	Concept	H-Index	Publications	Citations
1	Medicine	5	5	272
2	Engineering	4	4	133
3	Natural Sciences	4	4	227
4	Biochemistry	3	3	114
5	Biomolecular Engineering	3	3	120

Graham L. Simpson

Publications

673

Citations

H-Index

Page 1

	Year	Citations
Discovery and Characterization of a Cell-Permeable, Small-Molecule c-Abl Kinase Activator that Binds to the Myristoyl Binding Site Jingsong Yang, Nino Campobasso, Mangatt P. Biju, Chemistry & Biology Signal TransductionCell SignalingMyristoyl Binding SiteNatural SciencesMacromolecular Machine	2011	113
Design and Application of a DNA-Encoded Macrocyclic Peptide Library Zhengrong Zhu, Alex Shaginian, LaShadric C. Grady, ACS Chemical Biology	2017	103
Ladder Polyether Synthesis via Epoxide-Opening Cascades Using a Disappearing Directing Group Graham L. Simpson, Timothy P. Heffron, Estı́baliz Merino, Journal of the American Chemical Society Ladder Polyether SynthesisEngineeringTrimethylsilyl GroupMolecular BiologyOrganic Chemistry	2006	78
Improving the passive permeability of macrocyclic peptides: Balancing permeability with other physicochemical properties Praew Thansandote, Robert M. Harris, Hannah L. Dexter, Bioorganic & Medicinal Chemistry Peptide EngineeringPeptide LibraryPeptide SynthesisMembrane PermeationBalancing Permeability	2014	64
Synthesis and Pharmacological Characterization of Novel Analogues of the Nicotinic Acetylcholine Receptor Agonist (±)-UB-165 Christopher G. V. Sharples, Gunter Karig, Graham L. Simpson, Journal of Medicinal Chemistry Pharmacological CharacterizationNovel AnaloguesChemical BiologyExperimental PharmacologyMolecular Pharmacology	2002	52
Glycosylated Foldamers To Probe the Carbohydrate−Carbohydrate Interaction Graham L. Simpson, Andrew H. Gordon, David M. Lindsay, Journal of the American Chemical Society	2006	49
Intracellular drug concentration and disposition – The missing link? Michael M. Hann, Graham L. Simpson Methods PharmacodynamicsMedicinePhysiologyIntracellular Drug ConcentrationCellular Pharmacology	2014	43
The Discovery of in Vivo Active Mitochondrial Branched-Chain Aminotransferase (BCATm) Inhibitors by Hybridizing Fragment and HTS Hits Sophie M. Bertrand, Nicolas Ancellin, Benjamin Beaufils, Journal of Medicinal Chemistry Ligand EfficiencyMolecular BiologyPharmacotherapyHts HitsChemical Biology	2015	42
Ladder Polyether Synthesis via Epoxide-Opening Cascades Directed by a Disappearing Trimethylsilyl Group Timothy P. Heffron, Graham L. Simpson, Estı́baliz Merino, The Journal of Organic Chemistry	2010	30
Identification and Optimization of Novel Small c-Abl Kinase Activators Using Fragment and HTS Methodologies Graham L. Simpson, Sophie M. Bertrand, Alan D. Borthwick, Journal of Medicinal Chemistry	2019	28

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