Andrzej Kieltyka

Design and Synthesis of [(2,3-Dichlorophenyl)piperazin-1-yl]alkylfluorenylcarboxamides as Novel Ligands Selective for the Dopamine D₃Receptor Subtype

Michael J. Robarge, Stephen M. Husbands, Andrzej Kieltyka et al. · Journal of Medicinal Chemistry · 2001 · 86 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

Indoline and piperazine containing derivatives as a novel class of mixed D2/D4 receptor antagonists. Part 2: Asymmetric synthesis and biological evaluation

He Zhao, Xiao‐Shu He, Andrew Thurkauf et al. · Bioorganic & Medicinal Chemistry Letters · 2002 · 56 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +13

Design, synthesis, and discovery of 3-piperazinyl-3,4-dihydro-2(1H)-quinolinone derivatives

He Zhao, Andrew Thurkauf, Julia Braun et al. · Bioorganic & Medicinal Chemistry Letters · 2000 · 40 citations · Full text

Pharmacy, Chemistry, Medicinal Chemistry +10

<i>trans</i>-1-[(2-Phenylcyclopropyl)methyl]-4-arylpiperazines:  Mixed Dopamine D₂/D₄ Receptor Antagonists as Potential Antipsychotic Agents

Xiaoyan Zhang, Kevin J. Hodgetts, He Zhao et al. · Journal of Medicinal Chemistry · 2000 · 36 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

3-Aryl pyrazolo[4,3-d]pyrimidine derivatives

Jun Yuan, Michael Gulianello, Stéphane De Lombaert et al. · Bioorganic & Medicinal Chemistry Letters · 2002 · 34 citations · Full text