Livia Tepshi

Development of Thioaryl-Based Matrix Metalloproteinase-12 Inhibitors with Alternative Zinc-Binding Groups: Synthesis, Potentiometric, NMR, and Crystallographic Studies

Elisa Nuti, Doretta Cuffaro, E. Bernardini et al. · Journal of Medicinal Chemistry · 2018 · 71 citations · Full text

Pharmacy, Chemistry, Medicinal Chemistry +17

Mambalgin-1 Pain-relieving Peptide, Stepwise Solid-phase Synthesis, Crystal Structure, and Functional Domain for Acid-sensing Ion Channel 1a Inhibition

Gilles Mourier, Miguel Salinas, Pascal Kessler et al. · Journal of Biological Chemistry · 2015 · 66 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

Functional dissection of the retrograde Shiga toxin trafficking inhibitor Retro-2

Alison Forrester, Stefan Rathjen, Maria Daniela Garcia-Castillo et al. · Nature Chemical Biology · 2020 · 56 citations · Full text

Life Sciences, Cell Biology, Molecular Biology +13

Discovery of a new selective inhibitor of A Disintegrin And Metalloprotease 10 (ADAM-10) able to reduce the shedding of NKG2D ligands in Hodgkin's lymphoma cell models

Caterina Camodeca, Elisa Nuti, Livia Tepshi et al. · European Journal of Medicinal Chemistry · 2016 · 51 citations · Full text

Medicine, Medicinal Chemistry, Oncology +12

Sugar‐Based Arylsulfonamide Carboxylates as Selective and Water‐Soluble Matrix Metalloproteinase‐12 Inhibitors

Elisa Nuti, Doretta Cuffaro, Felicia D’Andrea et al. · ChemMedChem · 2016 · 50 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +12