Doug H. Falls

trans-Activation and Repression Properties of the Novel Nonsteroid Glucocorticoid Receptor Ligand 2,5-Dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5-(1-methylcyclohexen-3-y1)-1H-[1]benzopyrano[3,4-f]quinoline (A276575) and Its Four Stereoisomers

Chun Wel Lin, Masaki Nakane, Mike Stashko et al. · Molecular Pharmacology · 2002 · 50 citations

Life Sciences, Medicinal Chemistry, Pharmacology +17

Optimization of Chromone-2-carboxamide Melanin Concentrating Hormone Receptor 1 Antagonists:  Assessment of Potency, Efficacy, and Cardiovascular Safety

Jennifer C. Freeman, Andrew S. Judd, Rajesh Iyengar et al. · Journal of Medicinal Chemistry · 2006 · 48 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +13

Discovery and Characterization of Aminopiperidinecoumarin Melanin Concentrating Hormone Receptor 1 Antagonists

Philip R. Kym, Rajesh Iyengar, Andrew J. Souers et al. · Journal of Medicinal Chemistry · 2005 · 48 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +16

Aminopiperidine indazoles as orally efficacious melanin concentrating hormone receptor-1 antagonists

Anil Vasudevan, Andrew J. Souers, Jennifer C. Freeman et al. · Bioorganic & Medicinal Chemistry Letters · 2005 · 34 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +8

Identification of aminopiperidine benzamides as MCHr1 antagonists

Anil Vasudevan, Mary K. Verzal, Derek Wodka et al. · Bioorganic & Medicinal Chemistry Letters · 2005 · 15 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +7