Rien De Wachter

Synthesis of 4-amino-3-oxo-tetrahydroazepino[3,4-b]indoles: new conformationally constrained Trp analogs

Karolina Pulka‐Ziach, Debby Feytens, Isabelle Van den Eynde et al. · Tetrahedron · 2006 · 27 citations

Pharmacy, Medicinal Chemistry, Pharmacology +10

Conformationally constrained opioid ligands: The Dmt-Aba and Dmt-Aia versus Dmt-Tic scaffold

Steven Ballet, Debby Feytens, Rien De Wachter et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 25 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +11

Synthesis and Evaluation of the β‐Turn Properties of 4‐Amino‐1,2,4,5‐tetrahydro‐2‐benzazepin‐3‐ones and of Their Spirocyclic Derivative

Karolien Van Rompaey, Steven Ballet, Csaba Tömböly et al. · European Journal of Organic Chemistry · 2006 · 24 citations

Pharmacy, Chemistry, Medicinal Chemistry +9

Synthesis, Biological Evaluation, and Automated Docking of Constrained Analogues of the Opioid Peptide H-Dmt-<scp>d</scp>-Ala-Phe-Gly-NH₂Using the 4- or 5-Methyl Substituted 4-Amino-1,2,4,5-tetrahydro-2-benzazepin-3-one Scaffold

Rien De Wachter, Chris de Graaf, Atilla Keresztes et al. · Journal of Medicinal Chemistry · 2011 · 15 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Influence of ring substitution on the conformation and β-turn mimicry of 4-amino-1,2,4,5-tetrahydro-2-benzazepin-3-one peptide mimetics

Rien De Wachter, Luc Brans, Steven Ballet et al. · Tetrahedron · 2009 · 15 citations

Natural Sciences, Medicinal Chemistry, Pharmacology +14