Stéphane Ciblat

Discovery and Characterization of SY-1365, a Selective, Covalent Inhibitor of CDK7

Shanhu Hu, Jason Marineau, Nisha Rajagopal et al. · Cancer Research · 2019 · 146 citations

Discovery of SY-5609: A Selective, Noncovalent Inhibitor of CDK7

Jason Marineau, Kristin B. Hamman, Shanhu Hu et al. · Journal of Medicinal Chemistry · 2021 · 80 citations · Full text

Identification of <b>RP-6685</b>, an Orally Bioavailable Compound that Inhibits the DNA Polymerase Activity of Polθ

Monica Bubenik, P. Mäder, Philippe Mochirian et al. · Journal of Medicinal Chemistry · 2022 · 61 citations · Full text

Tetrahydrofuran-Based Transient Receptor Potential Ankyrin 1 (TRPA1) Antagonists: Ligand-Based Discovery, Activity in a Rodent Asthma Model, and Mechanism-of-Action via Cryogenic Electron Microscopy

Jack A. Terrett, Huifen Chen, Daniel G. Shore et al. · Journal of Medicinal Chemistry · 2021 · 49 citations · Full text

A simple and efficient enantioselective synthesis of piperidine alkaloids dihydropinidine and isosolenopsins A, B and C

Stéphane Ciblat, P. Besse-Hoggan Besse-Hoggan Pascale Pascale Besse, Vassiliki Papastergiou et al. · Tetrahedron Asymmetry · 2000 · 44 citations

Enantioselective Synthesis, Bioorganic Chemistry, Medicine +8